|
T6641 |
Rilmenidine Phosphate
|
|
Apoptosis
,
Adrenergic Receptor
,
Autophagy
,
Imidazoline Receptor
|
|
Rilmenidine Phosphate is a selective I(1) imidazoline receptor agonist, used to treat hypertension. |
|
T22051 |
BU 224 hydrochloride
|
|
Imidazoline Receptor
|
|
BU 224 hydrochloride is a selective imidazoline I(2) binding site ligand and has antinociceptive and antidepressant-like activities. |
|
T0115 |
Idazoxan hydrochloride
|
RX 781094 |
Adrenergic Receptor
,
Imidazoline Receptor
|
|
Idazoxan hydrochloride (RX 781094) is a benzodioxane-linked imidazole. It has alpha-2 adrenoceptor antagonist activity. |
|
T22052 |
BU 226 hydrochloride
|
|
Imidazoline Receptor
|
|
BU 226 hydrochloride demonstrates affinity for imidazoline (I) receptors, in particular the I2 binding site with a Ki of 1.4 nM. BU 226 hydrochloride showed low (microM) affinity for alpha 2-adrenoceptors. |
|
T1028 |
Moxonidine
|
BDF5895 |
Imidazoline Receptor
|
|
Moxonidine (BDF5895) is a selective agonist at the imidazoline receptor subtype 1, acting as an antihypertensive drug. |
|
T15010 |
CR4056
|
6-(1H-imidazol-1-yl)-2-phenylquinazoline |
MAO
,
Imidazoline Receptor
|
|
CR4056 (6-(1H-imidazol-1-yl)-2-phenylquinazoline) is a selective inhibitor of MAO-A with IC50 of 202.7 nM and a ligand of I2-imidazoline receptor with IC50 of 596 nM. |
|
T23283 |
2-Methoxyidazoxan monohydrochloride
|
RX 821002 hydrochloride |
Adrenergic Receptor
|
|
L-Albizziin (2-Methoxyidazoxan monohydrochloride) is a highly potent selective antagonist of the alpha 2r adrenergic receptor, with little or no antagonistic effect on imidazoline. It has a significantly higher affinity ... |
|
T6703 |
Tetrahydrozoline hydrochloride
|
Murine Plus,Tetryzoline hydrochloride,Tyzine,Tetrahydrozoline HCl |
Adrenergic Receptor
|
|
Tetrahydrozoline hydrochloride (Murine Plus) is an imidazoline derivative with alpha receptor agonist activity. |
|
T22492 |
2-BFI hydrochloride
|
|
Imidazoline Receptor
|
|
2-BFI hydrochloride is a high-affinity agonist of I2-imidazoline receptor. 2-BFI hydrochloride can be used in studies about protection against stroke and acute inflammatory immune disease. |
|
T21911 |
Rilmenidine hemifumarate
|
Rilmenidine (hemifumarate),S-3341 hemifumarate |
Apoptosis
,
Imidazoline Receptor
|
|
Rilmenidine hemifumarate (S-3341 hemifumarate) is a novel, orally active and selective I1 imidazoline receptor and α2-adrenoceptor agonist that induces autophagy, regulates the proliferation of leukaemia cells, stimulate... |
|
T23263 |
RS 45041-190 hydrochloride
|
|
Others
|
|
Highly selective I2 imidazoline receptor ligand |
|
T22760 |
Efaroxan hydrochloride
|
|
Others
|
|
α2 adrenoceptor antagonist and imidazoline I1 receptor ligand |
|
T26171 |
S23757
|
S-23757,S 23757 |
|
|
S23757 is an imidazoline 1 receptor (I1R) selective ligand. |
|
T68931 |
Tracizoline
|
|
|
|
Tracizoline is a potent I2-imidazoline receptor agonist. |
|
T40869 |
Moxonidine hydrochloride
|
BDF5895hydrochloride |
|
|
Moxonidine Hydrochloride serves as a selective agonist for the imidazoline receptor subtype 1 and functions as an antihypertensive agent. It primarily acts within the central nervous system and demonstrates a significant... |
|
T27155 |
Dexisometheptene
|
TNX 201,TNX-201,(R)-Isometheptene,TNX201 |
|
|
Dexisometheptene is an antimigraine drug candidate. Dexisometheptene significantly increases the pain threshold of acute pain response, and potently and selectively binds to receptors in the central nervous system known ... |
|
T73214 |
RX 801077
|
2 BFI free base |
|
|
RX 801077 (2 BFI free base), a selective imidazoline I2 receptor (I2R) agonist, exhibits a K i value of 70.1 nM, demonstrating anti-inflammatory and neuroprotective properties. This compound holds research potential for ... |
|
T35591 |
Guanfacine-13C,15N3
|
Guanfacine-13C,15N3 |
|
|
Guanfacine-13C,15N3is intended for us as an internal standard for the quantification of guanfacine by GC- or LC-MS. Guanfacine is an α2-adrenergic receptor (α2-AR) agonist with Kivalues of 93, 1,380, and 3,890 nM for α2A... |
